Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50036935
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  0.200nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataKi:  4.80nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100125(3-Isopropyl-4-methyl-pent-2-enoic acid 3-hydroxy-2...)
Affinity DataKi:  24.6nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50087241(3-Isopropyl-4-methyl-pentanoic acid (S)-1-hydroxym...)
Affinity DataKi:  28.6nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100126(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  31.1nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50015677((S)-1-hydroxymethyl-2-octanoyloxy-ethyl ester | 1,...)
Affinity DataKi:  33nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100129(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxy-2-(3...)
Affinity DataKi:  39.9nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100122(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  44.5nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100118(CHEMBL59422 | Octadec-9-enoic acid 2-acetoxy-3-hyd...)
Affinity DataKi:  50.4nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100127(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  68.3nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100123(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxy-2-(3...)
Affinity DataKi:  71nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100119(3-Isopropyl-4-methyl-pent-2-enoic acid 3-hydroxy-2...)
Affinity DataKi:  73nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100115(3-Isopropyl-4-methyl-pentanoic acid 1-hydroxymethy...)
Affinity DataKi:  74.9nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50087240((E)-Octadec-9-enoic acid (S)-1-hydroxymethyl-2-((E...)
Affinity DataKi:  87.2nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100117(3-Isopropyl-4-methyl-pent-2-enoic acid 3-hydroxy-2...)
Affinity DataKi:  110nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100120(3-Isopropyl-4-methyl-pentanoic acid 1-hydroxymethy...)
Affinity DataKi:  154nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100121(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  330nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100116(3-Methyl-but-2-enoic acid 1-hydroxymethyl-2-(3-met...)
Affinity DataKi:  1.05E+3nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100128(3-Methyl-butyric acid 1-hydroxymethyl-2-(3-methyl-...)
Affinity DataKi:  1.41E+3nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100124(3-Methyl-but-2-enoic acid 3-hydroxy-2-(3-methyl-bu...)
Affinity DataKi:  1.80E+3nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50100113(3-Methyl-but-2-enoic acid 1-hydroxymethyl-2-(3-met...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed