Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type' and Ligand = 'BDBM50087241'
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50087241(3-Isopropyl-4-methyl-pentanoic acid (S)-1-hydroxym...)
Affinity DataKi:  28.6nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087241(3-Isopropyl-4-methyl-pentanoic acid (S)-1-hydroxym...)
Affinity DataKi:  29nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087241(3-Isopropyl-4-methyl-pentanoic acid (S)-1-hydroxym...)
Affinity DataKi:  29nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed