Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50014227
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of the compound against human growth hormone secretagogue (GHS) receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139789(CHEMBL353389 | {3-[2-(3-Bromo-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of the compound against human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  28nMAssay Description:Inhibition of the compound against human angiotensin II receptor, type 1 (AG2-R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50049481((R)-N-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)meth...)
Affinity DataIC50:  60nMAssay Description:Inhibition of the compound against rat growth hormone secretagogue (GHS) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Sus scrofa)
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Curated by ChEMBL
LigandPNGBDBM50049481((R)-N-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)meth...)
Affinity DataIC50:  63nMAssay Description:Inhibition of the compound against pig growth hormone secretagogue (GHS) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139791(CHEMBL353007 | MC4 ligand)
Affinity DataIC50:  100nMAssay Description:Inhibition of the compound against human melanocortin-4 (MC4) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139791(CHEMBL353007 | MC4 ligand)
Affinity DataIC50:  190nMAssay Description:Inhibition of the compound against human growth hormone secretagogue (GHS) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139790(CHEMBL170530 | {5-[2-(4-Bromo-phenyl)-5-methyl-1H-...)
Affinity DataIC50:  612nMAssay Description:Inhibition of the compound against human melanocortin-4 (MC4) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50049481((R)-N-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)meth...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of the compound against human growth hormone secretagogue (GHS) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50049481((R)-N-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)meth...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of the compound against human angiotensin II receptor, type 1 (AG2-R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed