Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 1504
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50:  20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11820((3R,4R)-N-(4-{4-[5-(3,3-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50:  23nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50:  30nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11821((3R,4R)-N-(4-{4-[5-(4,4-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  40nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50:  400nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11818((3R,4R)-N-(4-{4-[3-(3,3-dimethylpiperidin-2-yl)-2-...)
Affinity DataIC50:  750nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11821((3R,4R)-N-(4-{4-[5-(4,4-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  1.70E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11820((3R,4R)-N-(4-{4-[5-(3,3-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  1.90E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11818((3R,4R)-N-(4-{4-[3-(3,3-dimethylpiperidin-2-yl)-2-...)
Affinity DataIC50:  2.40E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB