BDBM11817 (3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)benzoylamino]azepan-3-yl}isonicotinamide hydrochloride::N-[(3R,4R)-4-[(4-{[5-(dimethylamino)-2-hydroxyphenyl]carbonyl}benzene)amido]azepan-3-yl]pyridine-4-carboxamide hydrochloride::Protein Kinase B-Selective Inhibitor 1
SMILES CN(C)c1ccc(O)c(c1)C(=O)c1ccc(cc1)C(=O)N[C@@H]1CCCNC[C@H]1NC(=O)c1ccncc1
InChI Key InChIKey=NYQLXXDGJNYPPH-DNQXCXABSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 11817
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Max-Planck-Institut Fuer Biochemie
Max-Planck-Institut Fuer Biochemie
Affinity DataIC50: 30nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie
Max-Planck-Institut Fuer Biochemie
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair