Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50016473
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149275(2-(1-benzyl-5-(4-(trifluoromethoxy)phenyl)-1H-indo...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169448(1-Benzyl-3-phenyl-5-(4-trifluoromethoxy-benzenesul...)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169451(1-Biphenyl-4-ylmethyl-5-(4-tert-butyl-phenylamino)...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149274(2-[4-(3,4-Dichloro-phenylcarbamoyl)-benzylamino]-4...)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169446(1-Benzyl-5-(biphenyl-4-sulfonylamino)-3-phenyl-1H-...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169450(5-Benzenesulfonylamino-1-biphenyl-4-ylmethyl-3-phe...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169447(1-Benzyl-5-(4-tert-butyl-benzenesulfonylamino)-3-p...)
Affinity DataIC50:  2.87E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169449(1-Benzyl-5-(biphenyl-4-sulfonylamino)-1H-indole-2-...)
Affinity DataIC50:  6.31E+4nMAssay Description:Inhibitory concentration against Plasminogen activator inhibitor-1 by antibody assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed