Compile Data Set for Download or QSAR
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Found 74 Enz. Inhib. hit(s) with all data for entry = 5540
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86965((S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86964(2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4...)
Affinity DataKi:  0.470nMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86968((S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86969((R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86981((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86961((S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86974((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86978((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  2.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86969((R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86974((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86260(CAS_465-65-6 | NALOXONE | NSC_10064 | Naloxone(-))
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86963((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86962((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86961((S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl...)
Affinity DataKi:  8.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86260(CAS_465-65-6 | NALOXONE | NSC_10064 | Naloxone(-))
Affinity DataKi:  9.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86963((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86975((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86983((S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyph...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86964(2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4...)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86972((S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyp...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86983((S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyph...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86981((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86977((S)-2-(N-ethyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-...)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86958((S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)...)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86969((R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86966((S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydro...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86980((S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4...)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86972((S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyp...)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86971((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86971((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86978((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86970((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86260(CAS_465-65-6 | NALOXONE | NSC_10064 | Naloxone(-))
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86979((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  36nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86980((S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4...)
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
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Curated by PDSP Ki Database
LigandPNGBDBM86960((S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydrox...)
Affinity DataKi:  52nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86982((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  58nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86973((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86959((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86973((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86970((S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl...)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86969((R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86960((S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydrox...)
Affinity DataKi:  74nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86967((S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phe...)
Affinity DataKi:  80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86978((S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dim...)
Affinity DataKi:  83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86964(2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86966((S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydro...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86961((S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl...)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86967((S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phe...)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by PDSP Ki Database
LigandPNGBDBM86958((S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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