Compile Data Set for Download or QSAR
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Found 22 Enz. Inhib. hit(s) with all data for entry = 50043097
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKi:  11nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKi:  185nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKi:  1.98E+3nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKi:  1.50E+4nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKi:  1.54E+4nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  135nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436039(CHEMBL2392185)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 using SAPATGGVK(Me2)KPHRYRPGTVAL as substrate incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 using SAPATGGVK(Me2)KPHRYRPGTVAL as substrate incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  1.40E+3nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436039(CHEMBL2392185)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of JMJD2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50361475(CHEMBL1938900)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant 6xHis-tagged JMJD3 (unknown origin) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50361475(CHEMBL1938900)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of JMJD2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436039(CHEMBL2392185)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of recombinant 6xHis-tagged JMJD3 (unknown origin) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant 6xHis-tagged JMJD3 (unknown origin) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  1.45E+4nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of JMJD2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  1.09E+5nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataIC50:  1.12E+5nMAssay Description:Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKd:  19nMAssay Description:Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKd:  22nMAssay Description:Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Colorado

Curated by ChEMBL
LigandPNGBDBM50436040(CHEMBL2392184)
Affinity DataKd:  8.20nMAssay Description:Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed