Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 6343
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM50277889(CARFILZOMIB | CHEMBL451887)
Affinity DataIC50:  8.60nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
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TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  8.96nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM123812(4-Fluoro-N-{3-{S-4-methyl-1-[S-4-methyl-1-(R-2-met...)
Affinity DataIC50:  970nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM123813(4-Methoxy-N-{3-{S-4-methyl-1-[S-4-methyl-1-(R-2-me...)
Affinity DataIC50:  1.01E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM123811(N-{3-{S-4-Methyl-1-[S-4-methyl-1-(R-2-methyloxiran...)
Affinity DataIC50:  1.42E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM123810(N-{3-{S-4-Methyl-1-[S-4-methyl-1-(R-2-methyloxiran...)
Affinity DataIC50:  1.85E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed