Found 30 Enz. Inhib. hit(s) with all data for entry = 50047725 
Affinity DataKi: 0.143nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.367nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.458nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.875nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 381nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 472nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 573nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 2.36E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 4.23E+3nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 4.67E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University
Curated by ChEMBL
Nanjing Medical University
Curated by ChEMBL
Affinity DataKi: 1.92E+4nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 254nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 755nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 781nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 7.17E+3nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
