Affinity DataKi: 2.36E+3nMAssay Description:Binding affinity of the compound against delta-opioid receptor by using [3H]-DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.92E+4nMAssay Description:Binding affinity to DOP (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.92E+4nMAssay Description:Binding affinity against opioid receptor delta by displacement of radioligand [3H]-DSLET in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.92E+4nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 781nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair