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Found 35 Enz. Inhib. hit(s) with all data for entry = 50048955
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231393(CHEMBL4073167)
Affinity DataKi:  72nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to MCL1 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231393(CHEMBL4073167)
Affinity DataKi:  260nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  440nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to MCL1 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231392(CHEMBL4086474)
Affinity DataKi:  490nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to MCL1 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231391(CHEMBL4098080)
Affinity DataKi:  530nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to MCL1 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231390(CHEMBL4069319)
Affinity DataKi:  600nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to MCL1 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231393(CHEMBL4073167)
Affinity DataKi:  710nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl-XL (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231392(CHEMBL4086474)
Affinity DataKi:  740nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231391(CHEMBL4098080)
Affinity DataKi:  750nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  760nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  810nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl-XL (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231402(CHEMBL4073739)
Affinity DataKi:  910nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231390(CHEMBL4069319)
Affinity DataKi:  920nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231405(CHEMBL4064581)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231392(CHEMBL4086474)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl-XL (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231404(CHEMBL4061809)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231461(CHEMBL4105118)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231390(CHEMBL4069319)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl-XL (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231509(CHEMBL4099537)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231508(CHEMBL4065151)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231506(CHEMBL4102087)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231505(CHEMBL4080049)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231469(CHEMBL4090357)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231468(CHEMBL4074232)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231467(CHEMBL4075795)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231466(CHEMBL4088176)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231462(CHEMBL4094740)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231510(CHEMBL4100020)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231401(CHEMBL4086589)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231399(CHEMBL4064104)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231398(CHEMBL4091860)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231397(CHEMBL4084099)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231395(CHEMBL4097046)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231394(CHEMBL4061309)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50231403(CHEMBL4094340)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of N-terminal FAM-labeled Bid-BH3 peptide binding to Bcl2 (unknown origin) preincubated for 30 mins followed by N-terminal FAM-labeled Bid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed