Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50043431
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50441090(CHEMBL2430323 | US9669028, 114 N-(3-(3-methyl-1H-p...)
Affinity DataIC50:  233nMAssay Description:Inhibition of human CHK1 in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50229971(4-(4-(2,3-Dihydrobenzo[1,4]dioxin-6-yl)-5-pyridin-...)
Affinity DataIC50:  353nMAssay Description:Inhibition of rat CK1delta in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50441090(CHEMBL2430323 | US9669028, 114 N-(3-(3-methyl-1H-p...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human ERK8 in presence of 5 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50441089(CHEMBL2430324)
Affinity DataIC50:  838nMAssay Description:Inhibition of rat CK1delta in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50441090(CHEMBL2430323 | US9669028, 114 N-(3-(3-methyl-1H-p...)
Affinity DataIC50:  894nMAssay Description:Inhibition of rat CK1delta in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of Edinburgh Cancer Research Centre In The Institute Of Genetics And Molecular Medicine

Curated by ChEMBL
LigandPNGBDBM50441090(CHEMBL2430323 | US9669028, 114 N-(3-(3-methyl-1H-p...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human NEK2alpha in presence of 50 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed