Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50036288
TargetGastrin/cholecystokinin type B receptor(RAT)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataEC50:  1.00E+3nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataKd:  1.40nMAssay Description:Tested in vitro by the gastrin binding assay for the competitive binding with iodinated gastrin for the gastrin receptors in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50037875(CBS-4 | CHEMBL341330)
Affinity DataEC50:  130nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50037874(CBS-5 | CHEMBL124944)
Affinity DataEC50:  80nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50037873(CBS-2 | CHEMBL341130)
Affinity DataEC50:  2.00E+5nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataKd:  3.20nMAssay Description:Tested in vitro for gastrin binding to gastrin receptors from guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed