Reaction Details Report a problem with these data
Target
Somatostatin receptor type 4
Ligand
BDBM84627
Substrate
n/a
Ki
15±n/a nM
Comments
PDSP_394
Citation
 Raynor, K; O'Carroll, AM; Kong, H; Yasuda, K; Mahan, LC; Bell, GI; Reisine, T Characterization of cloned somatostatin receptors SSTR4 and SSTR5. Mol Pharmacol 44:385-92 (1993) [PubMed] 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SSR4_RAT | Somatostatin receptor | Somatostatin receptor type 4 | Sstr4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42096.84
Organism:
RAT
Description:
SOMATOSTATIN SST4 SSTR4 RAT::P30937
Residue:
384
Sequence:
MNTPATLPLGGEDTTWTPGINASWAPDEEEDAVRSDGTGTAGMVTIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASAAALRHWPFGAVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAVFADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGPGCICPPLPCQQEPMQAEPACKRVPFTKTTTF
  
Inhibitor
Name:
BDBM84627
Synonyms:
BIM 23067
Type:
Small organic molecule
Emp. Form.:
C56H72ClN11O9
Mol. Mass.:
1078.692
SMILES:
CC[C@H](NC(=O)[C@H](N)Cc1ccc(Cl)cc1)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C)C(=O)N[C@H](Cc1ccccc1)C(N)=O
Structure:
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