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Found 501 with Last Name = 'kong' and Initial = 'h'
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82463(Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*hepta...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82552(CAS_111555-58-9 | NTB | naltrindolebenzofuran)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50039022(4-[(S)-((2R,5S)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442922(CHEMBL3086984)
Affinity DataKi:  0.0310nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442927(CHEMBL3086994)
Affinity DataKi:  0.0320nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442921(CHEMBL3086985)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442924(CHEMBL3086982)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442930(CHEMBL3086991)
Affinity DataKi:  0.0490nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442926(CHEMBL3086995)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82555(CAS_4424 | NSC_4424 | Naloxonazine)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50382474(CHEMBL2024096 | US9303017, Sazetidine-A)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442928(CHEMBL3086993)
Affinity DataKi:  0.0720nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442920(CHEMBL3086986)
Affinity DataKi:  0.0760nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50013388(6-Ethyl-3-(1-hydroxy-cyclopropylmethyl)-11,11-dime...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82462(BIM 23059 | D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82427(CAS_5985-38-6 | LEVORPHANOL-tartarate)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82554(Beta C N A | CAS_115070 | NSC_115070)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442929(CHEMBL3086992)
Affinity DataKi:  0.0830nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442923(CHEMBL3086983)
Affinity DataKi:  0.0930nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442932(CHEMBL3086989)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50169774(2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50166908(5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50072110(3-((S)-1-Azetidin-2-ylmethoxy)-5-phenyl-pyridine |...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50019574(CHEMBL406014 | CTOP | D-Phe-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM21865((14beta)-17-(cyclopropylmethyl)-18-(1-hydroxy-1-me...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(RAT)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50442925(CHEMBL3086996)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR after 4 hrs by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82553(BETA-FUNALTREXAMINE | CAS_72786-10-8 | b-FNA-HCl)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82550(CAS_118476-87-2 | Dermorphin | NSC_125954)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
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