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Target
Granzyme K
Ligand
BDBM50187800
Substrate
n/a
Meas. Tech.
ChEMBL_385595 (CHEMBL869128)
Ki
>150000±n/a nM
Citation
Sperandio, D; Tai, VW; Lohman, J; Hirschbein, B; Mendonca, R; Lee, CS; Spencer, JR; Janc, J; Nguyen, M; Beltman, J; Sprengeler, P; Scheerens, H; Lin, T; Liu, L; Gadre, A; Kellogg, A; Green, MJ; McGrath, ME Novel, potent, selective, and orally bioavailable human betaII-tryptase inhibitors. Bioorg Med Chem Lett 16:4085-9 (2006) [PubMed] Article
More Info.:
Target
Name:
Granzyme K
Synonyms:
Fragmentin-3 | GRAK_HUMAN | GZMK | Granzyme-3 | NK-TRYP-2 | NK-tryptase-2 | TRYP2
Type:
PROTEIN
Mol. Mass.:
28902.79
Organism:
Homo sapiens (Human)
Description:
ChEMBL_162618
Residue:
264
Sequence:
MTKFSSFSLFFLIVGAYMTHVCFNMEIIGGKEVSPHSRPFMASIQYGGHHVCGGVLIDPQWVLTAAHCQYRFTKGQSPTVVLGAHSLSKNEASKQTLEIKKFIPFSRVTSDPQSNDIMLVKLQTAAKLNKHVKMLHIRSKTSLRSGTKCKVTGWGATDPDSLRPSDTLREVTVTVLSRKLCNSQSYYNGDPFITKDMVCAGDAKGQKDSCKGDSGGPLICKGVFHAIVSGGHECGVATKPGIYTLLTKKYQTWIKSNLVPPHTN