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TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50539421(CHEMBL4634355)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate incubated for 20 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  2.30nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405397(CHEMBL2051983)
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024137(1-Hydroxymethyl-5-(2-hydroxy-2-phenyl-ethylamino)-...)
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024119(5-(2-Hydroxy-cyclohexylamino)-1-hydroxymethyl-cycl...)
Affinity DataIC50: 6.10nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  10nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024124(1-Hydroxymethyl-5-(2-hydroxy-1-phenyl-ethylamino)-...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50226273(CHEMBL3349431)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50327503((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  15nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50637820(CHEMBL5555649)
Affinity DataIC50: 20nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-alpha-D-glucopyranoside as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50330961((2R,3S,4S)-1-((2S,3S,4R,5R,6S)-2,3,4,5,6,7-hexahyd...)
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  28nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405395(CHEMBL2051761)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50330954(de-O-sulfonated kotalanol | CHEMBL1276973)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50259956(2,6-Bis-hydroxymethyl-piperidine-3,4,5-triol | alp...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity measured against alpha-glucosidase of rice by colorimetric assay using the D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 40nMAssay Description:Inhibitory concentration against human alpha-glucosidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50327502((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  43nMAssay Description:Inhibition of human N-terminal maltase-glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024136(5-(3,5-Di-tert-butyl-4-hydroxy-benzylamino)-1-hydr...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50327502((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  50nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50330960((2R,3R,4R)-1-((2R,3R,4S,5R,6S)-2,3,4,5,6,7-hexahyd...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405396(CHEMBL2051762)
Affinity DataIC50: 68nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405389(CHEMBL2051982)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  70nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405393(CHEMBL2051981)
Affinity DataIC50: 72nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50611854(CHEMBL5271914)
Affinity DataIC50: 77nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50330959(CHEMBL1277153)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50613821(CHEMBL4854113)
Affinity DataIC50: 82nMAssay Description:Inhibition of alpha glucosidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50611832(CHEMBL4856778)
Affinity DataIC50: 85nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  87nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50316180((2S,3S,4R,5S,6S)-1-((2R,3S,4S)-3,4-dihydroxy-2-(hy...)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50405387(CHEMBL2051759)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024139(1-Hydroxymethyl-5-phenethylamino-cyclohexane-1,2,3...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Glycosidases (maltase) in rat intestinal brush border membranes by D-glucose oxidase-peroxidase method maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50613819(CHEMBL3944972)
Affinity DataIC50: 120nMAssay Description:Inhibition of alpha glucosidase (unknown origin) using p-nitrophenyl glucopyranoside as substrate pre incubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50316181((2S,3S,4R,5S,6R)-1-((2R,3S,4S)-3,4-dihydroxy-2-(hy...)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50: 150nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50327501(ponkoranol | CHEMBL1258528)
Affinity DataKi:  170nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50: 172nMAssay Description:Inhibition of alpha glucosidase (unknown origin) using p-nitrophenyl glucopyranoside as substrate by UV Vis- spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50613820(CHEMBL4855744)
Affinity DataIC50: 186nMAssay Description:Inhibition of alpha glucosidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024116(1-Hydroxymethyl-5-(2-hydroxy-2-phenyl-ethylamino)-...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024120(1-Hydroxymethyl-5-[(thiophen-2-ylmethyl)-amino]-cy...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50614755(CHEMBL5271502)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of Alpha-glucosidase (unknown origin) by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50316178(1,4-Dideoxy-1,4-[[2S,3S,4R,5R,6R-2,4,5,6,7-pentahy...)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetMaltase-glucoamylase(Human)
University of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50024128(5-(4-Bromo-benzylamino)-1-hydroxymethyl-cyclohexan...)
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
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