Compile Data Set for Download or QSAR
Report error Found 151 of affinity data for UniProtKB/TrEMBL: P09487
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068225(CHEMBL3403324)
Affinity DataKi:  50nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068229(CHEMBL3403327)
Affinity DataKi:  60nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50428400([(4-Methylphenyl)Sulfonyl]Phenylamine | CHEMBL1826...)
Affinity DataKi:  70nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50165140(CHEMBL3797297)
Affinity DataKi:  78nMAssay Description:Inhibition of bovine tissue non-specific alkaline phosphatase preincubated for 3 to 5 mins followed by CDP-star substrate addition measured after 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222186(6-(Dimethylamino)-3-(4'-nitrophenyl)-2,3-dihyd...)
Affinity DataIC50: 110nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222186(6-(Dimethylamino)-3-(4'-nitrophenyl)-2,3-dihyd...)
Affinity DataIC50: 110nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068225(CHEMBL3403324)
Affinity DataIC50: 115nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068230(CHEMBL3403329)
Affinity DataKi:  128nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50437935(CHEMBL2408701)
Affinity DataKi:  130nMAssay Description:Inhibition of bovine kidney intestinal alkaline phosphatase using p-NPP as substrate treated 10 mins before substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068229(CHEMBL3403327)
Affinity DataIC50: 150nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50428400([(4-Methylphenyl)Sulfonyl]Phenylamine | CHEMBL1826...)
Affinity DataIC50: 180nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50165140(CHEMBL3797297)
Affinity DataIC50: 180nMAssay Description:Inhibition of bovine tissue non-specific alkaline phosphatase preincubated for 3 to 5 mins followed by CDP-star substrate addition measured after 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222179(6-(Dimethylamino)-3-phenyl-2,3-dihydronaphtho[1,8-...)
Affinity DataIC50: 190nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222179(6-(Dimethylamino)-3-phenyl-2,3-dihydronaphtho[1,8-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222188(6-(Dimethylamino)-3-(4'-hydroxy-3'-methoxy...)
Affinity DataIC50: 200nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222188(6-(Dimethylamino)-3-(4'-hydroxy-3'-methoxy...)
Affinity DataIC50: 200nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50437931(CHEMBL2408705)
Affinity DataKi:  250nMAssay Description:Inhibition of bovine kidney intestinal alkaline phosphatase using p-NPP as substrate treated 10 mins before substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222189(6-(Dimethylamino)-3-(3'-hydroxy-4'-methoxy...)
Affinity DataIC50: 270nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222189(6-(Dimethylamino)-3-(3'-hydroxy-4'-methoxy...)
Affinity DataIC50: 270nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222185(6-(Dimethylamino)-3-(3',5'-dichloro-2-hydr...)
Affinity DataIC50: 270nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222185(6-(Dimethylamino)-3-(3',5'-dichloro-2-hydr...)
Affinity DataIC50: 270nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068220(CHEMBL3403320)
Affinity DataKi:  299nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222190(6-(Dimethylamino)-3-(3'-bromo-4'-methoxyph...)
Affinity DataIC50: 300nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222190(6-(Dimethylamino)-3-(3'-bromo-4'-methoxyph...)
Affinity DataIC50: 300nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222187(6-(Dimethylamino)-3-(2'-methoxyphenyl)-2,3-dih...)
Affinity DataIC50: 310nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068230(CHEMBL3403329)
Affinity DataIC50: 310nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222187(6-(Dimethylamino)-3-(2'-methoxyphenyl)-2,3-dih...)
Affinity DataIC50: 310nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM223077((E)-N'-(4'-Hydroxy-3-methoxybenzylidene)is...)
Affinity DataIC50: 350nMpH: 9.8 T: 2°CAssay Description:The assay conditions were optimized with some changes in formerly reported spectrophotometric method. The composition of assay buffer of pH 9.8 was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222180(6-(Dimethylamino)-3-(4'-dichlorophenyl)-2,3-di...)
Affinity DataIC50: 420nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222180(6-(Dimethylamino)-3-(4'-dichlorophenyl)-2,3-di...)
Affinity DataIC50: 420nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222191(6-(Dimethylamino)-3-(5'-bromo-2'-hydroxy-3...)
Affinity DataIC50: 440nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222191(6-(Dimethylamino)-3-(5'-bromo-2'-hydroxy-3...)
Affinity DataIC50: 440nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222181(6-(Dimethylamino)-3-(4'-methylphenyl)-2,3-dihy...)
Affinity DataIC50: 460nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222181(6-(Dimethylamino)-3-(4'-methylphenyl)-2,3-dihy...)
Affinity DataIC50: 460nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222182(6-(Dimethylamino)-3-(4'-hydroxyphenyl)-2,3-dih...)
Affinity DataIC50: 500nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222182(6-(Dimethylamino)-3-(4'-hydroxyphenyl)-2,3-dih...)
Affinity DataIC50: 500nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222192(6-(Dimethylamino)-3-(2',3',4'-trimetho...)
Affinity DataIC50: 510nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM223074((E)-N'-(4'-Methoxybenzylidene)isonicotinoh...)
Affinity DataIC50: 560nMpH: 9.8 T: 2°CAssay Description:The assay conditions were optimized with some changes in formerly reported spectrophotometric method. The composition of assay buffer of pH 9.8 was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068220(CHEMBL3403320)
Affinity DataIC50: 613nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50165131(CHEMBL3797468)
Affinity DataKi:  623nMAssay Description:Inhibition of bovine tissue non-specific alkaline phosphatase preincubated for 3 to 5 mins followed by CDP-star substrate addition measured after 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222191(6-(Dimethylamino)-3-(5'-bromo-2'-hydroxy-3...)
Affinity DataIC50: 680nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068228(CHEMBL3403317)
Affinity DataKi:  918nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50068227(CHEMBL3403325)
Affinity DataKi:  950nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM223080((E)-N'-(1-(3-(4-fluorophenyl)-5-phenyl-4,5-dih...)
Affinity DataIC50: 1.06E+3nMpH: 9.8 T: 2°CAssay Description:The assay conditions were optimized with some changes in formerly reported spectrophotometric method. The composition of assay buffer of pH 9.8 was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222192(6-(Dimethylamino)-3-(2',3',4'-trimetho...)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated with enzyme for 3 to 5 mins followed by substrate addition and measured after 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222192(6-(Dimethylamino)-3-(2',3',4'-trimetho...)
Affinity DataIC50: 1.19E+3nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50247721(4-fluoro-N-(4-sulfamoylbenzyl)benzenesulfonamide |...)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM50234702(CHEMBL4066927)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of bovine TNAP using CDP-star as substrate preincubated for 5 to 7 mins followed by substrate addition measured after 15 mins by spectroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2019
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM16661(1-N-(4-fluorobenzene)benzene-1,4-disulfonamide | a...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of bovine kidney non-specific alkaline phosphatase using CDP-star chemiluminescent substrate assessed as change in luminescence by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2016
Entry Details Article
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Bovine)
Forman Christian College (A Chartered University)

Curated by ChEMBL
LigandPNGBDBM222184(6-(Dimethylamino)-3-(3'-nitrophenyl)-2,3-dihyd...)
Affinity DataIC50: 1.45E+3nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2017
Entry Details Article
PubMed
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