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TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476140(CHEMBL373632)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85009(H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2018
Entry Details

TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476137(CHEMBL222751)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85009(H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214421(SOMATOSTATIN RECEPTOR LIGAND)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82466(L-362862 | c[Aha-Phe-p-C1-Phe-D-Trp-Lys-Thr-Phe] |...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85229(BIM 23295)
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476135(CHEMBL374316)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.860nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50272772(CHEMBL1680 | 10-(4-Amino-butyl)-19-(2-amino-3-phen...)
Affinity DataIC50: 1nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059093(2-{[10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propio...)
Affinity DataIC50: 1.04nMAssay Description:Compound was tested for the inhibition of rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82457((1R,4S,7S,10R,13S,16R)-4-[(R)-1-Hydroxyethyl]-7-(4...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059091(2-{[9-(4-Amino-butyl)-18-(2-amino-3-phenyl-propion...)
Affinity DataIC50: 1.29nMAssay Description:Compound was tested for the inhibition of rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059091(2-{[9-(4-Amino-butyl)-18-(2-amino-3-phenyl-propion...)
Affinity DataIC50: 1.30nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476143(CHEMBL376001)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  1.58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85011(AcNH-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85012(AcNH-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKi:  3.23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82468(D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-D-Phe-NH2 | BIM 23...)
Affinity DataKi:  3.31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82456(CAS_117580-24-2 | BIM 23030)
Affinity DataKi:  3.89nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  4.46nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82467(CGP-23996 | 2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-...)
Affinity DataKi:  4.67nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
Affinity DataKi:  5.49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059089(9-(4-Amino-butyl)-18-(2-amino-3-phenyl-propionylam...)
Affinity DataIC50: 5.5nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059089(9-(4-Amino-butyl)-18-(2-amino-3-phenyl-propionylam...)
Affinity DataIC50: 5.5nMAssay Description:Compound was tested for the inhibition of rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82461(D-Phe-AIa-Tyr-D-Trp-Lys-Val-Ala-D-Nal-NH2 | BIM 23...)
Affinity DataKi:  5.88nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82455(BIM-23027 | N-Methylcyclo[L-Ala-L-Tyr-D-Trp-L-Lys-...)
Affinity DataKi:  6.16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  8.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85230(BIM 23313)
Affinity DataKi:  9.88nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059092((4S,7R,10S,13R,16S,19R)-10-(4-Amino-butyl)-19-((S)...)
Affinity DataIC50: 10.6nMAssay Description:Compound was tested for the inhibition of rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50059092((4S,7R,10S,13R,16S,19R)-10-(4-Amino-butyl)-19-((S)...)
Affinity DataIC50: 11nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
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