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TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.0800nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311957(US10166214, Example 93 | US9789082, Example 93 | U...)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311970(US10166214, Example 106 | US10675268, Example 106)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474230(CHEMBL3349516)
Affinity DataKi: <0.100nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311957(US10166214, Example 93 | US9789082, Example 93 | U...)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50597579(CHEMBL5197201)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311970(US10166214, Example 106 | US10675268, Example 106)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM506557(US11045457, Example 157)
Affinity DataEC50:  0.126nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM506589(US11045457, Example 190)
Affinity DataEC50:  0.158nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474219(CHEMBL3349522)
Affinity DataKi: <0.200nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474221(CHEMBL3349521)
Affinity DataKi: <0.200nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50597589(CHEMBL5209180)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.200nMAssay Description:Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476134(CHEMBL437296)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311971(US10166214, Example 107 | US9789082, Example 107 |...)
Affinity DataEC50:  0.200nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM523757(US11136312, Compound MM-I-87)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311971(US10166214, Example 107 | US9789082, Example 107 |...)
Affinity DataEC50:  0.200nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311973(US10166214, Example 109 | US10675268, Example 109)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM312007(US10166214, Example 143 | US10675268, Example 143)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311944(US10166214, Example 80 | US9789082, Example 80 | U...)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM312007(US10166214, Example 143 | US10675268, Example 143)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50597576(CHEMBL5180543)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311967(US10166214, Example 103 | US10675268, Example 103)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311944(US10166214, Example 80 | US9789082, Example 80 | U...)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311973(US10166214, Example 109 | US10675268, Example 109)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311967(US10166214, Example 103 | US10675268, Example 103)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311994(US10166214, Example 130 | US10675268, Example 130)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311994(US10166214, Example 130 | US10675268, Example 130)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM523756(US11136312, Compound MM-I-83)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50474231(CHEMBL3349513)
Affinity DataKi: <0.316nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82547(SRIF-D-Trp8)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476138(CHEMBL376485)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM506615(US11045457, Example 216)
Affinity DataEC50:  0.398nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50081055(CHEMBL3421843 | US10166214, Example 49 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human somatostatin 4 receptor expressed in H4 cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM312048(US10166214, Example 184 | US10675268, Example 184)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50081055(CHEMBL3421843 | US10166214, Example 49 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50081058(CHEMBL3421842 | US10166214, Example 22 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50081055(CHEMBL3421843 | US10166214, Example 49 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311969(US10166214, Example 105 | US10675268, Example 105)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311939(US10166214, Example 75 | US10675268, Example 75)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311939(US10166214, Example 75 | US10675268, Example 75)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM311969(US10166214, Example 105 | US10675268, Example 105)
Affinity DataEC50:  0.400nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

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