Compile Data Set for Download or QSAR
Report error Found 59 of affinity data for UniProtKB/TrEMBL: P32198
LigandChemical structure of BindingDB Monomer ID 50024430BDBM50024430((R) (R) -2-Tetradecyl-oxirane-2-carboxylic acid-Co...)
Affinity DataIC50: 20nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50024434BDBM50024434((+/-) 2-Tetradecyl-oxirane-2-carboxylic acid-Coenz...)
Affinity DataIC50: 30nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50024432BDBM50024432((R)-(+)2-Tetradecyl-oxirane-2-carboxylic acid | CH...)
Affinity DataIC50: 30nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50024431BDBM50024431((+/-)2-Tetradecyl-oxirane-2-carboxylic acid | 2-Te...)
Affinity DataIC50: 40nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50024429BDBM50024429((R)-(+)2-Tetradecyl-oxirane-2-carboxylic acid meth...)
Affinity DataIC50: 40nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50024433BDBM50024433(2-Tetradecyl-oxirane-2-carboxylic acid methyl este...)
Affinity DataIC50: 90nMAssay Description:Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122836BDBM50122836([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataKi:  360nMAssay Description:Inhibition of rat liver carnitine palmitoyltransferase IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101604BDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 700nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101598BDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 700nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50403029BDBM50403029(CHEMBL2216792)
Affinity DataIC50: 700nMAssay Description:Inhibition of rat CPT1A expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101591BDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101591BDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 800nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50403040BDBM50403040(CHEMBL2216779)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of rat hepatocytes CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50240113BDBM50240113(CHEMBL4081425)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat wild-type CPT1A expressed in yeast mitochondrial extracts using L-[methyl-3H]carnitine and palmitoyl-CoA as substrates preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122839BDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50403039BDBM50403039(CHEMBL2216778)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of rat hepatocytes CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50101594BDBM50101594([3-Carboxy-2-(decane-1-sulfonylamino)-propyl]-trim...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122834BDBM50122834([3-Carboxy-2-(3-dodecyl-ureido)-propyl]-trimethyl-...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101589BDBM50101589([3-Carboxy-2-(nonylaminosulphonyl-amino)-propyl]-t...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50639700BDBM50639700(CHEMBL5561479)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to rat heart mitochondria CPT1 assessed as inhibition constant incubated for 3 to 6 mins by Liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50122828BDBM50122828([3-Carboxy-2-(3-undecyl-ureido)-propyl]-trimethyl-...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50033117BDBM50033117([3-Carboxy-2-(hydroxy-tetradecyloxy-phosphoryloxy)...)
Affinity DataKi:  3.60E+3nMAssay Description:In vitro inhibition of carnitine palmitoyltransferase I with respect to palmitoyl CoA in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50046145BDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataKi:  4.20E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50639700BDBM50639700(CHEMBL5561479)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to rat liver mitochondria CPT1 assessed as inhibition constant incubated for 3 to 6 mins by Liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50101604BDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101600BDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101598BDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101600BDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122833BDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50403046BDBM50403046(CHEMBL2216772)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50240112BDBM50240112(CHEMBL4099442)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of rat wild-type CPT1A expressed in yeast mitochondrial extracts using L-[methyl-3H]carnitine and palmitoyl-CoA as substrates preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101590BDBM50101590([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101593BDBM50101593((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122827BDBM50122827([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50046145BDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataIC50: 3.85E+4nMAssay Description:Inhibition of rat CPT1A using [3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50046145BDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataIC50: 3.85E+4nMAssay Description:Inhibition of rat CPT1A using [3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122837BDBM50122837([3-Carboxy-2-(3-heptyl-ureido)-propyl]-trimethyl-a...)
Affinity DataIC50: 4.36E+4nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101597BDBM50101597((3-Carboxy-2-tetradecyloxy-propyl)-trimethyl-ammon...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122836BDBM50122836([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 61402BDBM61402(perhexiline maleate | (Z)-but-2-enedioic acid;2-(2...)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of CPT1 in rat cardiac mitochondria using [3H]carnitine by radiometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101607BDBM50101607([3-Carboxy-2-(3-nonyl-thioureido)-propyl]-trimethy...)
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50284163BDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibitory potency against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50117921BDBM50117921(2-(2,2-dicyclohexylethyl)piperidine | Perhexilene ...)
Affinity DataIC50: 1.48E+5nMAssay Description:Inhibition of rat CPT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 61402BDBM61402(perhexiline maleate | (Z)-but-2-enedioic acid;2-(2...)
Affinity DataIC50: 1.48E+5nMAssay Description:Inhibition of CPT1 in rat liver mitochondria using [3H]carnitine by radiometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101608BDBM50101608((3-Carboxy-2-tetradecylamino-propyl)-trimethyl-amm...)
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22984BDBM22984(Adriamycin | (8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of rat CPT1 in rat mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101602BDBM50101602(1-(2-Nonylcarbamoyloxy-3-phosphono-propyl)-pyridin...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101601BDBM50101601((3-Carboxy-2-octyloxy-propyl)-trimethyl-ammonium |...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101603BDBM50101603((3-Carboxy-2-octylamino-propyl)-trimethyl-ammonium...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50101592BDBM50101592((3-Carboxy-2-nonylcarbamoyloxy-propyl)-trimethyl-a...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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