Compile Data Set for Download or QSAR
Report error Found 1298 of affinity data for UniProtKB/TrEMBL: P47900
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045627BDBM50045627(US9540323, 200 | CHEMBL3314307 | US9540323, exampl...)
Affinity DataIC50: 0.0200nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045625BDBM50045625(US9540323, 198 | CHEMBL3314305 | US9540323, exampl...)
Affinity DataIC50: 0.0300nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017084BDBM50017084(CHEMBL3287050 | US9428504, 61)
Affinity DataIC50: 0.0300nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045628BDBM50045628(US9540323, 202 | CHEMBL3314308 | US9540323, exampl...)
Affinity DataIC50: 0.0400nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017089BDBM50017089(CHEMBL3287043 | US9428504, 8)
Affinity DataIC50: 0.0400nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017090BDBM50017090(CHEMBL3287044 | US9428504, 59)
Affinity DataIC50: 0.0400nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045611BDBM50045611(US9540323, 77 | CHEMBL3314291 | US9540323, example...)
Affinity DataIC50: 0.0500nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017083BDBM50017083(CHEMBL3287049 | US9428504, 39)
Affinity DataIC50: 0.0600nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045626BDBM50045626(US9540323, 201 | CHEMBL3314306 | US9540323, exampl...)
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015286BDBM50015286(CHEMBL3263066 | US9120798, 3)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017085BDBM50017085(CHEMBL3287051 | US9428504, 60)
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045610BDBM50045610(US9540323, 74 | CHEMBL3314290 | US9540323, example...)
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045606BDBM50045606(CHEMBL3314320 | US9428504, 155)
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015276BDBM50015276(CHEMBL3263056 | US9428504, 166 | US9428504, 167)
Affinity DataIC50: 0.120nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045597BDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human P2Y1 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045597BDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50: 0.120nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015276BDBM50015276(CHEMBL3263056 | US9428504, 166 | US9428504, 167)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045597BDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50: 0.120nMAssay Description:Antagonist activity at human P2Y1 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015276BDBM50015276(CHEMBL3263056 | US9428504, 166 | US9428504, 167)
Affinity DataIC50: 0.120nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017088BDBM50017088(CHEMBL3287042 | US9428504, 89)
Affinity DataIC50: 0.130nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045624BDBM50045624(US9540323, 209 | CHEMBL3314304 | US9540323, exampl...)
Affinity DataIC50: 0.130nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045619BDBM50045619(US9540323, 205 | CHEMBL3314299 | US9540323, exampl...)
Affinity DataIC50: 0.130nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017087BDBM50017087(CHEMBL3287041 | US9428504, 10)
Affinity DataIC50: 0.140nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045607BDBM50045607(CHEMBL3314287)
Affinity DataIC50: 0.140nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045615BDBM50045615(US9540323, 206 | CHEMBL3314297 | US9540323, exampl...)
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017086BDBM50017086(CHEMBL3287052 | US9428504, 79)
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045605BDBM50045605(CHEMBL3314319 | US9428504, 157)
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017075BDBM50017075(CHEMBL3287040 | US9428504, 38)
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015277BDBM50015277(CHEMBL3263057 | US9120798, 1)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015296BDBM50015296(CHEMBL3263076 | US9120798, 13)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015287BDBM50015287(CHEMBL3263067 | US9120798, 2)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045629BDBM50045629(US9540323, 194 | CHEMBL3314309 | US9540323, exampl...)
Affinity DataIC50: 0.230nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017021BDBM50017021(CHEMBL3287047 | US9428504, 1)
Affinity DataIC50: 0.230nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045604BDBM50045604(US9540323, 164 | CHEMBL3314317 | US9540323, exampl...)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015289BDBM50015289(CHEMBL3263069 | US9120798, 44)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045617BDBM50045617(US9540323, 193 | CHEMBL3314298 | US9540323, exampl...)
Affinity DataIC50: 0.330nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015288BDBM50015288(CHEMBL3263068 | US9120798, 46)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045613BDBM50045613(US9540323, 207 | CHEMBL3314296 | US9540323, exampl...)
Affinity DataIC50: 0.370nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045612BDBM50045612(US9540323, 195 | CHEMBL3314295 | US9540323, exampl...)
Affinity DataIC50: 0.370nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017091BDBM50017091(CHEMBL3287045 | US9428504, 6)
Affinity DataIC50: 0.370nMAssay Description:Antagonist activity at P2Y1 receptor in human platelets by FLIPR assay in presence of 2-methylthio-ADPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045608BDBM50045608(US9540323, 56 | CHEMBL3314288 | US9540323, example...)
Affinity DataIC50: 0.390nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409523BDBM50409523(CHEMBL2112093)
Affinity DataEC50:  0.400nMAssay Description:Accumulation of inositol phosphate in 1321N1 astrocytoma cells expressing human P2Y1 purinoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409523BDBM50409523(CHEMBL2112093)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human P2Y1R in human 1321N1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045631BDBM50045631(US9540323, 232 | CHEMBL3314310 | US9540323, exampl...)
Affinity DataIC50: 0.450nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045603BDBM50045603(US9540323, 161 | CHEMBL3314316 | US9540323, exampl...)
Affinity DataIC50: 0.470nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045601BDBM50045601(US9540323, 135 | CHEMBL3314315 | US9540323, exampl...)
Affinity DataIC50: 0.510nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045621BDBM50045621(US9540323, 203 | CHEMBL3314301 | US9540323, exampl...)
Affinity DataIC50: 0.520nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045600BDBM50045600(US9540323, 149 | CHEMBL3314314 | US9540323, exampl...)
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045623BDBM50045623(US9540323, 197 | CHEMBL3314303 | US9540323, exampl...)
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015291BDBM50015291(CHEMBL3263071 | US9120798, 26)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of P2Y1 receptor in human washed platelets assessed as decrease in 2-methylthio-ADP-induced calcium signal transduction pathway activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
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