Compile Data Set for Download or QSAR
Report error Found 487 of affinity data for UniProtKB/TrEMBL: P48145
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603459(CHEMBL5187335)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603429(CHEMBL5170622)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603433(CHEMBL5204006)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603467(CHEMBL5197385)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 5.90nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50: 6nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50013388(CHEMBL350384 | BREMAZOCINE(-) | 6-Ethyl-3-(1-hydro...)
In Depth
Date in BDB:
12/21/2011
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603459(CHEMBL5187335)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603429(CHEMBL5170622)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603428(CHEMBL5194519)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603446(CHEMBL5178929)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603430(CHEMBL5172042)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603431(CHEMBL5206425)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603469(CHEMBL5177662)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50: 18nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603468(CHEMBL5188323)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50: 21nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603475(CHEMBL5179908)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603432(CHEMBL5191528)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603433(CHEMBL5204006)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603467(CHEMBL5197385)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50553728(CHEMBL4757321)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50553728(CHEMBL4757321)
Affinity DataIC50: 30nMAssay Description:Negative allosteric modulation activity at NPBWR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50: 35nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603471(CHEMBL5208352)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603442(CHEMBL5174290)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50553729(CHEMBL4796786)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603455(CHEMBL5189212)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603472(CHEMBL5195844)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603470(CHEMBL5194208)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50553730(CHEMBL4779758)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603458(CHEMBL5196275)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603447(CHEMBL5185639)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50247803(Beta-Funeltrexamine | beta-funaltrexamine | methyl...)
Affinity DataKi:  93nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2011
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50: 95nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603457(CHEMBL5200286)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50425599(CHEMBL2314291)
Affinity DataIC50: 100nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603461(CHEMBL5191389)
Affinity DataEC50:  112nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603462(CHEMBL5198182)
Affinity DataIC50: 113nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50425598(CHEMBL1972527)
Affinity DataIC50: 120nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50425597(CHEMBL2314320)
Affinity DataIC50: 140nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | Tyr-Pro-Phe-Pro-NH2 | [D-Pro4]morph...)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2011
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50401576(CHEMBL2207117)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603449(CHEMBL5180015)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
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