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Report error Found 14 of affinity data for UniProtKB/TrEMBL: P62744
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  18nMAssay Description:Binding affinity to human AP2S1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  24.2nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339687(4-(Dimethylamino)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339689(4-(2-Fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)-piper...)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  678nMAssay Description:Binding affinity to human AP2S1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339686(4-(2-Fluoroethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phen...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339688(4-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339683(4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339691(4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  1.57E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339684(4-(2-Fluoroethyl)-N-(4-(4-(2-(2-Fluoroethoxy)pheny...)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339690(4-(2-fluoroethyl)-N-(4-(4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  2.21E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50339685(4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  5.96E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM81790(NSC_2159 | CAS_71675-85-9 | Amisulpride | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed