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Report error Found 992 of affinity data for UniProtKB/TrEMBL: Q07912
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621875BDBM50621875(CHEMBL5400397)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421256BDBM50421256(CHEMBL2087874)
Affinity DataKi:  0.200nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421257BDBM50421257(CHEMBL2087875)
Affinity DataKi:  0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621877BDBM50621877(CHEMBL5408748)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421256BDBM50421256(CHEMBL2087874)
Affinity DataKi:  0.300nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2016
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421255BDBM50421255(CHEMBL2087873)
Affinity DataKi:  0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621883BDBM50621883(CHEMBL5431206)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621855BDBM50621855(CHEMBL5409024)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621858BDBM50621858(CHEMBL5398945)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621888BDBM50621888(CHEMBL5419830)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621880BDBM50621880(CHEMBL5428907)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621878BDBM50621878(CHEMBL5405674)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621884BDBM50621884(CHEMBL5399309)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621876BDBM50621876(CHEMBL5437496)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621882BDBM50621882(CHEMBL5439245)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419721BDBM419721(US10464919, Example 59)
Affinity DataIC50: 0.920nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419799BDBM419799(US10464919, Example 137)
Affinity DataIC50: 0.950nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13216BDBM13216(N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyeth...)
Affinity DataIC50: 1nMAssay Description:Inhibition of ACK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204580BDBM50204580(N-phenethyl-5-phenyl-6-(4-(2-(pyrrolidin-1-yl)etho...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Ack1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621881BDBM50621881(CHEMBL5436567)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621879BDBM50621879(CHEMBL5434969)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419844BDBM419844(US10464919, Example 182)
Affinity DataIC50: 1.26nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621862BDBM50621862(CHEMBL5431312)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419794BDBM419794(US10464919, Example 132)
Affinity DataIC50: 1.31nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419731BDBM419731(US10464919, Example 69)
Affinity DataIC50: 1.32nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419781BDBM419781(US10464919, Example 119)
Affinity DataIC50: 1.38nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419751BDBM419751(US10464919, Example 89)
Affinity DataIC50: 1.48nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419791BDBM419791(US10464919, Example 129)
Affinity DataIC50: 1.65nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419758BDBM419758(US10464919, Example 96)
Affinity DataIC50: 1.75nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419797BDBM419797(US10464919, Example 135)
Affinity DataIC50: 1.75nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419740BDBM419740(US10464919, Example 78)
Affinity DataIC50: 1.87nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621871BDBM50621871(CHEMBL5404048)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419832BDBM419832(US10464919, Example 170)
Affinity DataIC50: 1.96nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419755BDBM419755(US10464919, Example 93)
Affinity DataIC50: 1.97nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419761BDBM419761(US10464919, Example 99)
Affinity DataIC50: 1.99nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245854BDBM50245854(N3-(2,6-dichlorophenyl)-N6-(3-fluoro-4-(2-(pyrroli...)
Affinity DataKi:  2nMAssay Description:Inhibition of histidine-tagged ACK1 (amino acids 117 to 489) expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421286BDBM50421286(CHEMBL2087662)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 482158BDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  2nMAssay Description:Binding constant for TNK2 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246162BDBM50246162(N3-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl...)
Affinity DataKi:  2nMAssay Description:Inhibition of histidine-tagged ACK1 (amino acids 117 to 489) expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421278BDBM50421278(CHEMBL2087654)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421276BDBM50421276(CHEMBL2087652)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246164BDBM50246164(N3-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl...)
Affinity DataIC50: 2nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2016
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337126BDBM50337126(US9266890, IV-2 | CHEMBL1672987 | Scaffold, B19 | ...)
Affinity DataKd:  2nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2016
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246214BDBM50246214(N3-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl...)
Affinity DataKi:  2nMAssay Description:Inhibition of histidine-tagged ACK1 (amino acids 117 to 489) expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621890BDBM50621890(CHEMBL5415503)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419765BDBM419765(US10464919, Example 103)
Affinity DataIC50: 2.10nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419842BDBM419842(US10464919, Example 180)
Affinity DataIC50: 2.12nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419784BDBM419784(US10464919, Example 122)
Affinity DataIC50: 2.37nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419785BDBM419785(US10464919, Example 123)
Affinity DataIC50: 2.38nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419804BDBM419804(US10464919, Example 142)
Affinity DataIC50: 2.45nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

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