TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 0.0180nMAssay Description:Inhibition of the GAR formyl transferase in L1210More data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of the GAR formyl transferase in L1210More data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKd: 0.25nMAssay Description:Thermodynamic dissociation constant (KD) was measured upon binding to GAR TFase in miceMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of GAR transformylase from Lactobacillus caseiMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of mouse recombinant GARFtase assessed as FGAR formation by spectrophotometryMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Tested for the inhibition against the human dihydrofolate reductaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:In vitro inhibition of mouse GAR transformylaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Compound was tested for inhibition constant against GAR TFase in miceMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Tested for the inhibition of trifunctional Glycinamide ribonucleotide formyltransferase isolated from murine L1210 cells.More data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 147nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of GAR transformylase from mammalian MancaMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of GAR transformylase from mammalian L1210 cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 710nMAssay Description:Inhibitory activity against murine glycinamide ribonucleotide formyltransferase (GARFT) enzymeMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of GAR transformylase from Lactobacillus caseiMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of mouse recombinant GARFtase assessed as FGAR formation by spectrophotometryMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:potent inhibitor of GAR Tfase obtained from porcineMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of mouse recombinant GARFtase assessed as FGAR formation by spectrophotometryMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 5.51E+3nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 8.52E+3nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Inhibitory activity against murine glycinamide ribonucleotide formyltransferase (GARFT) enzymeMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of GAR transformylase from mammalian MancaMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GAR transformylase from mammalian L1210 cellsMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GAR transformylase from Lactobacillus caseiMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GAR transformylase from Lactobacillus caseiMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GAR transformylase from mammalian MancaMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
University of South Alabama
Curated by ChEMBL
University of South Alabama
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse recombinant GARFTaseMore data for this Ligand-Target Pair












3D Structure (crystal)


























