Compile Data Set for Download or QSAR
Report error Found 4 of affinity data for UniProtKB/TrEMBL: Q7TNH1
TargetPeroxisome proliferator-activated receptor alpha(Golden hamster)
Bristol-Myers Squibb

LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  488nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Golden hamster)
Bristol-Myers Squibb

LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  178nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Golden hamster)
Bristol-Myers Squibb

LigandPNGBDBM28803(Clofop | HCG 004 | 2-[4-(4-chlorophenoxy)phenoxy]p...)
Affinity DataEC50:  2.87E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Golden hamster)
Bristol-Myers Squibb

LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  488nMAssay Description:Agonist activity at syrian golden hamster PPARalpha LBD (167-468) expressed in HEK293 cells coexpressing GAL4-DBD by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed