Compile Data Set for Download or QSAR
Report error Found 562 of affinity data for UniProtKB/TrEMBL: Q8R4B8
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605051BDBM50605051(CHEMBL5184952)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse BMDM cells assessed as reduction in ATP induced IL-1beta release pretreated for 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse BMDM cells assessed as reduction in ATP induced IL-1beta release pretreated for 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505850BDBM50505850(Dapansutrile | OLT-1177 | OLT1177)
Affinity DataIC50: 1nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774A.1 cells assessed as reduction in IL-1beta level preincubated for 30 mins follow...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505850BDBM50505850(Dapansutrile | OLT-1177 | OLT1177)
Affinity DataIC50: 1nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta level incubated for 1 hr followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50632650BDBM50632650(CHEMBL5421905)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-treated mouse BMDM cells assessed as inhibition of ATP-stimulated IL-1beta release incubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in LPS/ATP-treated mouse bone marrow derived macrophages assessed as reduction in NLRP3 inflammasome activation by measuring redu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse BMDM assessed as reduction in NLRP3 inflammasome-induced IL-1beta production prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDM cells preincubated for 30 mins followed by ATP addition by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDMsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDMsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in mouse BMDM preincubated with LPS for 3 hrs followed by compound addition for 30 mins and further stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse BMDM cells assessed as inhibition of LPS and nigericin-induced IL-1beta pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse bone marrow derived macrophages assessed as reduction in IL-1beta level preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50598221BDBM50598221(CHEMBL4288808)
Affinity DataIC50: 8nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50632651BDBM50632651(CHEMBL5422387)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-treated mouse BMDM cells assessed as inhibition of ATP-stimulated IL-1beta release incubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 13nMAssay Description:Inhibition of NLRP3 inflammasome in mouse JJ74.A1 cells assessed as inhibition of LPS/ATP-induced IL-1 beta release stimulated with LPS for 4.5 hs fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 14nMAssay Description:Inhibition of NLRP3 inflammasome in mouse JJ74.A1 cells assessed as inhibition of LPS/ATP-induced IL-1 beta secretion primed with LPS for 4.5 hs foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636753BDBM50636753(Emlenoflast | Inzomelid | Izd-174 | Izd174 | MCC-7...)
Affinity DataIC50: 14nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50634192BDBM50634192(CHEMBL5396485)
Affinity DataIC50: 14nMAssay Description:Inhibition of NLRP3 in mouse BMDM cells assessed as reduction in IL-1beta productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647995BDBM50647995(CHEMBL5597392)
Affinity DataIC50: 15nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin stimulated mouse BMDMs assessed as reduction in IL-1beta release pretreated with LPS for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636753BDBM50636753(Emlenoflast | Inzomelid | Izd-174 | Izd174 | MCC-7...)
Affinity DataIC50: 16nMAssay Description:Inhibition of NLRP3 in mouse BMDMs assessed as reduction in LPS/ATP-induced IL-1beta release preincubated for 30 mins in presence of LPS followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50632652BDBM50632652(CHEMBL5436366)
Affinity DataIC50: 20nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-treated mouse BMDM cells assessed as inhibition of ATP-stimulated IL-1beta release incubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 22nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 23nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse J774A.1 cells assessed as decrease in LDH release pretreated for 0.5 hrs f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 23nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse J774A.1 cells assessed as decrease in IL-1beta level pretreated for 0.5 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 761021BDBM761021(US20250243172, Compound Formula IV (YM-III-3))
Affinity DataKd:  24nMAssay Description:Monolith NT. Automated instrument was used to measure the Kd value. A range of concentrations of NSIs were incubated and His-NLRP3 pre-labeled with R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50652650BDBM50652650(CHEMBL5646860)
Affinity DataIC50: 24nMAssay Description:Inhibition of NLRP3 inflammasome-mediated IL-1beta release in LPS-primed neonatal C57BL/6 P1-4 mouse microglia pretreated for 30 mins followed by med...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622947BDBM50622947(CHEMBL5430191 | US20250243172, Compound Formula IX...)
Affinity DataKd:  25nMAssay Description:Monolith NT. Automated instrument was used to measure the Kd value. A range of concentrations of NSIs were incubated and His-NLRP3 pre-labeled with R...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50628782BDBM50628782(CHEMBL5434669)
Affinity DataIC50: 25nMAssay Description:Inhibition of NLRP3 inflammasome in mouse JJ74.A1 cells assessed as inhibition of LPS/ATP-induced IL-1 beta secretion primed with LPS for 4.5 hs foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622941BDBM50622941(CHEMBL5417338)
Affinity DataKd:  25nMAssay Description:Binding affinity to full-length mouse recombinant NLRP3 assessed as dissociation constant by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593017BDBM50593017(CHEMBL5196305)
Affinity DataIC50: 32nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 40nMAssay Description:Inhibition of NLRP3 in mouse peritoneal macrophages assessed as inhibition of LPS and ATP-induced IL-1beta production pre-stimulated with LPS for 4.5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 40nMAssay Description:Inhibition of NLRP3 in mouse peritoneal macrophages assessed as inhibition of LPS and ATP-induced IL-1beta production pre-stimulated with LPS for 4.5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069989BDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 41nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505855BDBM50505855(CHEMBL4468698)
Affinity DataIC50: 42nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse bone marrow derived macrophages assessed as reduction in IL-1beta level preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505855BDBM50505855(CHEMBL4468698)
Affinity DataIC50: 42nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-induced mouse BMDMs assessed as decrease in IL-1beta release preincubated for 30 mins followed by ATP additio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593025BDBM50593025(CHEMBL5187619)
Affinity DataIC50: 46nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593023BDBM50593023(CHEMBL5183504)
Affinity DataIC50: 49nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593013BDBM50593013(CHEMBL483266)
Affinity DataIC50: 49nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636758BDBM50636758(CHEMBL5561914)
Affinity DataIC50: 50nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607509BDBM50607509(CHEMBL5219789)
Affinity DataIC50: 63nMAssay Description:Inhibition of NLRP3 induced IL-1beta release in LPS/nigericin-treated mouse BMDM cells preincubated with LPS for 3 hrs followed by compound addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50628784BDBM50628784(CHEMBL5414644)
Affinity DataIC50: 63nMAssay Description:Inhibition of NLRP3 inflammasome in mouse JJ74.A1 cells assessed as inhibition of LPS/ATP-induced IL-1 beta secretion primed with LPS for 4.5 hs foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593016BDBM50593016(CHEMBL5195292)
Affinity DataIC50: 65nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622948BDBM50622948(CHEMBL5434916 | US20250243172, Compound Formula X ...)
Affinity DataKd:  69nMAssay Description:Monolith NT. Automated instrument was used to measure the Kd value. A range of concentrations of NSIs were incubated and His-NLRP3 pre-labeled with R...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636778BDBM50636778(CHEMBL5562815)
Affinity DataIC50: 72nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593018BDBM50593018(CHEMBL5171338)
Affinity DataIC50: 74nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593020BDBM50593020(CHEMBL5177370)
Affinity DataIC50: 76nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636762BDBM50636762(CHEMBL5567870)
Affinity DataIC50: 77nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Hospital Universitario Santa Cristina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593011BDBM50593011(CHEMBL5208208)
Affinity DataIC50: 79nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
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