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26 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and Evaluation of Diphenyl Conjugated Imidazole Derivatives as Potential Glutaminyl Cyclase Inhibitors for Treatment of Alzheimer's Disease.EBI
Shenzhen University
Discovery of Potent Human Glutaminyl Cyclase Inhibitors as Anti-Alzheimer's Agents Based on Rational Design.EBI
Seoul National University
Inhibitory effect of flavonoids on human glutaminyl cyclase.EBI
Shenzhen University
Structure-activity relationships of benzimidazole-based glutaminyl cyclase inhibitors featuring a heteroaryl scaffold.EBI
Probiodrug
Structure-activity relationship of human glutaminyl cyclase inhibitors having an N-(5-methyl-1H-imidazol-1-yl)propyl thiourea template.EBI
Seoul National University
Inhibitors for human glutaminyl cyclase by structure based design and bioisosteric replacement.EBI
Probiodrug
2-Amino-1,3,4-thiadiazoles as Glutaminyl Cyclases Inhibitors Increase Phagocytosis through Modification of CD47-SIRP? Checkpoint.EBI
Ewha Womans University
Discovery of highly potent human glutaminyl cyclase (QC) inhibitors as anti-Alzheimer's agents by the combination of pharmacophore-based and structure-based design.EBI
Seoul National University
Discovery of Conformationally Restricted Human Glutaminyl Cyclase Inhibitors as Potent Anti-Alzheimer's Agents by Structure-Based Design.EBI
Seoul National University
Potent human glutaminyl cyclase inhibitors as potential anti-Alzheimer's agents: Structure-activity relationship study of Arg-mimetic region.EBI
Seoul National University
Structure-activity relationship investigation of Phe-Arg mimetic region of human glutaminyl cyclase inhibitors.EBI
Seoul National University
Structural Origin of Selectivity in Class II-Selective Histone Deacetylase Inhibitors.BDB
University of Notre Dame
Development of potent purine-derived nitrile inhibitors of the trypanosomal protease TbcatB.BDB
University of California San Francisco
Pharmacophore analysis of the nuclear oxysterol receptor LXRalpha.BDB
Dartmouth College
N-Acylthiadiazolines, a new class of liver X receptor agonists with selectivity for LXRbeta.BDB
Gnf