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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Development of novel benzomorpholine class of diacylglycerol acyltransferase I inhibitors.EBI
Merck Research Laboratories
Irreversible inhibitors of cysteine proteases.EBI
Dart Neuroscience
Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI
University of Florida
Dipeptidyl aspartyl fluoromethylketones as potent caspase-3 inhibitors: SAR of the P2 amino acid.EBI
Maxim Pharmaceuticals
Structure-based discovery of a novel non-peptidic small molecular inhibitor of caspase-3.EBI
Tokyo University of Science
Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: peptidomimetic replacement of the P(2) amino acid by 2-aminoaryl acids and other non-natural amino acids.EBI
Epicept
Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: peptidomimetic replacement of the P2 alpha-amino acid by a alpha-hydroxy acid.EBI
Maxim Pharmaceuticals
Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: SAR of the N-protecting group.EBI
Maxim Pharmaceuticals
Oxamyl dipeptide caspase inhibitors developed for the treatment of stroke.EBI
Idun Pharmaceuticals
Quinolone hybrids and their anti-cancer activities: An overview.EBI
Qilu University of Technology (Shandong Academy of Sciences)
Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors.EBI
Roche Pharma Research and Early Development
Inhibitor of Apoptosis Protein (IAP) Antagonists in Anticancer Agent Discovery: Current Status and Perspectives.EBI
Ningxia Medical University
A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate.BDB
Whitehead Institute For Biomedical Research
Identification of 1, 4-Dihydrothieno [3', 2':5, 6]thiopyrano[4, 3-c] pyrazole derivatives as human 5-Lipo-oxygenase inhibitors.BDB
Peking University
Discovery of selective aminothiazole aurora kinase inhibitors.BDB
Novartis
Probing the elusive catalytic activity of vertebrate class IIa histone deacetylases.BDB
Irbm/Merck Research Laboratories