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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists.EBI
University of Regensburg
(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands.EBI
Jagiellonian University Medical College
Functional Profiling of 2-Aminopyrimidine Histamine H4 Receptor Modulators.EBI
Janssen Research and Development
Discovery and SAR of 6-alkyl-2,4-diaminopyrimidines as histamine H4 receptor antagonists.EBI
Janssen Research and Development
A novel series of histamine H4 receptor antagonists based on the pyrido[3,2-d]pyrimidine scaffold: comparison of hERG binding and target residence time with PF-3893787.EBI
Griffin Discoveries
Detailed structure-activity relationship of indolecarboxamides as H4 receptor ligands.EBI
Boehringer Ingelheim Rcv
Ligand based design of novel histamine H4 receptor antagonists; fragment optimization and analysis of binding kinetics.EBI
Griffin Discoveries
Challenges of drug discovery in novel target space. The discovery and evaluation of PF-3893787: a novel histamine H4 receptor antagonist.EBI
Pfizer
Agonist/antagonist modulation in a series of 2-aryl benzimidazole H4 receptor ligands.EBI
Johnson & Johnson Pharmaceutical Research & Development
Discovery of a Novel Highly Selective Histamine H4 Receptor Antagonist for the Treatment of Atopic Dermatitis.EBI
Sungkyunkwan University
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine HEBI
University of Regensburg
4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine HEBI
Vrije Universiteit Amsterdam
[EBI
University of Regensburg
Histamine H4 receptor agonists.EBI
University of Regensburg