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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of a highly potent, nonabsorbable apical sodium-dependent bile acid transporter inhibitor (GSK2330672) for treatment of type 2 diabetes.EBI
Glaxosmithkline
Expression and transport properties of the human ileal and renal sodium-dependent bile acid transporter.EBI
Wake Forest University
Identification of a region of the ileal-type sodium/bile acid cotransporter interacting with a competitive bile acid transport inhibitor.EBI
Ucla and The Wadsworth Veterans Administration Hospital
Discovery of potent, nonsystemic apical sodium-codependent bile acid transporter inhibitors (Part 2).EBI
Pfizer
Discovery of potent, nonsystemic apical sodium-codependent bile acid transporter inhibitors (Part 1).EBI
Pharmacia
Molecular switch controlling the binding of anionic bile acid conjugates to human apical sodium-dependent bile acid transporter.EBI
University of Maryland
Synthesis and biological evaluation of novel steroidal pyrazoles as substrates for bile acid transporters.EBI
Xenoport
A novel class of apical sodium-dependent bile acid transporter inhibitors: the amphiphilic 4-oxo-1-phenyl-1,4-dihydroquinoline derivatives.EBI
Sankyo
A novel class of apical sodium co-dependent bile acid transporter inhibitors: the 1,2-benzothiazepines.EBI
Pfizer
A novel class of apical sodium co-dependent bile acid transporter inhibitors: the 2,3-disubstituted-4-phenylquinolines.EBI
Searle Discovery
Design of Gut-Restricted Thiazolidine Agonists of G Protein-Coupled Bile Acid Receptor 1 (GPBAR1, TGR5).EBI
Ardelyx
Discovery of oxadiazoyl tertiary carbinamine inhibitors of beta-secretase (BACE-1).BDB
Merck Research Laboratories