Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50015524
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157077({(R)-4-[(4R,10aS,12aR)-4-Hydroxy-8-(2-hydroxy-ethy...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157075(2-[(4R)-4-[(2S,18R)-6-{2-[(6,7-dimethoxy-1,2,3,4-t...)
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157072({(R)-4-[(10aS,12aR)-8-(3-Hydroxy-benzyl)-10a,12a-d...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157079([(R)-4-((4R,10aS,12aR)-4-Hydroxy-10a,12a-dimethyl-...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157074({(R)-4-[(4R,10aS,12aR)-4-Hydroxy-8-(3-hydroxy-benz...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157076({(R)-4-[(10aS,12aR)-8-(2-Hydroxy-ethyl)-10a,12a-di...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157072({(R)-4-[(10aS,12aR)-8-(3-Hydroxy-benzyl)-10a,12a-d...)
Affinity DataIC50: 900nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157074({(R)-4-[(4R,10aS,12aR)-4-Hydroxy-8-(3-hydroxy-benz...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157078([(R)-4-((10aS,12aR)-10a,12a-Dimethyl-1,2,3,3a,3b,4...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157079([(R)-4-((4R,10aS,12aR)-4-Hydroxy-10a,12a-dimethyl-...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157080(2-[(4R)-4-[(2S,12R,18R)-12-hydroxy-6-[(3-{[(2S)-2-...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157081({(R)-4-[(4R,10aS,12S,12aR)-4,12-Dihydroxy-8-(3-hyd...)
Affinity DataIC50: 8.60E+3nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157077({(R)-4-[(4R,10aS,12aR)-4-Hydroxy-8-(2-hydroxy-ethy...)
Affinity DataIC50: 2.20E+4nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157075(2-[(4R)-4-[(2S,18R)-6-{2-[(6,7-dimethoxy-1,2,3,4-t...)
Affinity DataIC50: 3.20E+4nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157078([(R)-4-((10aS,12aR)-10a,12a-Dimethyl-1,2,3,3a,3b,4...)
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157073(2-[(4R)-4-[(2S,18R)-6-[(3-{[(2S)-2-(6-methoxynapht...)
Affinity DataIC50: 6.30E+4nMAssay Description:In vitro inhibition of taurocholate binding to liver bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157080(2-[(4R)-4-[(2S,12R,18R)-12-hydroxy-6-[(3-{[(2S)-2-...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157073(2-[(4R)-4-[(2S,18R)-6-[(3-{[(2S)-2-(6-methoxynapht...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157081({(R)-4-[(4R,10aS,12S,12aR)-4,12-Dihydroxy-8-(3-hyd...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Xenoport

Curated by ChEMBL
LigandPNGBDBM50157076({(R)-4-[(10aS,12aR)-8-(2-Hydroxy-ethyl)-10a,12a-di...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of taurocholate binding to human ileal bile acid transporter expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed