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27 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Development of Potent and Selective S. aureus Sortase A Inhibitors Based on Peptide Macrocycles.EBI
Ecole Polytechnique F�D�Rale De Lausanne
Discovery and structure-activity relationship studies of irreversible benzisothiazolinone-based inhibitors against Staphylococcus aureus sortase A transpeptidase.EBI
University of Latvia
Beta-carboline alkaloids derived from the ascidian Synoicum sp.EBI
Seoul National University
Discorhabdins from the Korean marine sponge Sceptrella sp.EBI
Seoul National University
Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform.EBI
M.V. Lomonosov Moscow State University
Activation of inhibitors by sortase triggers irreversible modification of the active site.EBI
University of Chicago
Identification of novel inhibitors of bacterial surface enzyme Staphylococcus aureus Sortase A.EBI
University of Alabama At Birmingham
Sesterterpenes from the tropical sponge Coscinoderma sp.EBI
Seoul National University
Synthetic analogs of indole-containing natural products as inhibitors of sortase A and isocitrate lyase.EBI
Institute
Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A Inhibitors.EBI
Nanjing University of Chinese Medicine
Chemical Biology of Sortase A Inhibition: A Gateway to Anti-infective Therapeutic Agents.EBI
Indian Institute of Technology Delhi
Antibacterial activity evaluation of vinyl sulfones against global predominant methicillin-resistant Staphylococcus aureus USA300.EBI
Mahidol University
Small Carbohydrate Derivatives as Potent Antibiofilm Agents.EBI
Indian Institute of Technology Bombay
Covalent sortase A inhibitor ML346 prevents EBI
Shanghai Institute of Materia Medica
Discovery of diarylacrylonitriles as a novel series of small molecule sortase A inhibitors.EBI
Seoul National University
Tideglusib and Its Analogues As Inhibitors of EBI
Guizhou University
Isocadiolides A-H: Polybrominated Aromatics from a EBI
Seoul National University
Pyrrolomycins as antimicrobial agents. Microwave-assisted organic synthesis and insights into their antimicrobial mechanism of action.EBI
University of Palermo
Discovery and development of substituted thiadiazoles as inhibitors of Staphylococcus aureus Sortase A.EBI
University of Gothenburg
Naturally Occurring Lumazines.EBI
University of Auckland
Synthetic small molecules as anti-biofilm agents in the struggle against antibiotic resistance.EBI
University of Palermo
Meroterpenoids from a Tropical Dysidea sp. Sponge.EBI
Seoul National University
Aaptamines as sortase A inhibitors from the tropical sponge Aaptos aaptos.EBI
Seoul National University
Bis(indole) alkaloids as sortase A inhibitors from the sponge Spongosorites sp.EBI
Seoul National University
Quinone skeleton as a new class of irreversible inhibitors against Staphylococcus aureus sortase A.EBI
Shanghai Institute of Materia Medica
Manzamine Alkaloids from an Acanthostrongylophora sp. Sponge.EBI
Seoul National University
Chemical compoundsBDB
Glaxosmithkline