Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50044783
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030337(CHEMBL3343843)
Affinity DataIC50: 3.39E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030335(CHEMBL3343842)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030322(CHEMBL3343832)
Affinity DataIC50: 3.81E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030321(CHEMBL3343831)
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030329(CHEMBL3343839)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030327(CHEMBL3343837)
Affinity DataIC50: 4.01E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030328(CHEMBL3343838)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030336(CHEMBL3341779)
Affinity DataIC50: 4.22E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030323(CHEMBL3343833)
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030320(CHEMBL3343830)
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030334(CHEMBL3343841)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030326(CHEMBL3343836)
Affinity DataIC50: 5.08E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM34709(SMR000154301 | cid_4875293 | N-(1-adamantyl)-2-(3-...)
Affinity DataIC50: 6.11E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030330(CHEMBL3343840)
Affinity DataIC50: 6.26E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030325(CHEMBL3343835)
Affinity DataIC50: 6.44E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030324(CHEMBL3343834)
Affinity DataIC50: 7.06E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50030338(CHEMBL3343844)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50201782(CHEMBL536752 | CHEMBL264166 | 1-(3,4-dichloropheny...)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Latvia

Curated by ChEMBL
LigandPNGBDBM50125084((ethenylsulfonyl)benzene | Ethenesulfonyl-benzene ...)
Affinity DataIC50: 7.36E+5nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed