BDBM129823 US8815926, 102

SMILES COc1ncc(-c2nc3C(=O)N([C@H](c3n2C(C)C)c2ccc(Cl)cc2)c2cc(Cl)cn(C)c2=O)c(OC)n1

InChI Key InChIKey=AGBSXNCBIWWLHD-FQEVSTJZSA-N

Data  1 KI  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 129823   

TargetProtein Mdm4(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM129823(US8815926, 102)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human MDM4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM129823(US8815926, 102)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of human MDM2 by TR-FRET assayMore data for this Ligand-Target Pair