BDBM50024418 5-Methyl-thiophene-2-carboxylic acid (3-imidazol-1-yl-propyl)-amide::CHEMBL8986

SMILES Cc1ccc(s1)C(=O)NCCCn1ccnc1

InChI Key InChIKey=ZMMSSWBMCUIDFQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50024418   

TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50024418(5-Methyl-thiophene-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human Nampt using NAM as substrate after 15 mins by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024418(5-Methyl-thiophene-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed