BDBM808428 7- (cyclopropylmeth- yl)-3-(2-{[(3S)- 6,6- dimethylpiperidin- 3-yl]amino}-5- (trifluoromethyl)py- rimidin-4-yl)- 1H,4H,5H,6H,7H, 8H-pyrrolo[2,3- c]azepin-8-one::US20260137698, Compound CDK7-1227
SMILES CC1(C)CC[C@H](Nc2ncc(C(F)(F)F)c(-c3c[nH]c4c3CCCN(CC3CC3)C4=O)n2)CN1
InChI Key InChIKey=BGGNKFVCLAAQKR-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 808428
Affinity DataIC50: 10nMAssay Description:Compounds were added to a 384-well plate. Reaction mixtures contained 10 mM HEPES, pH 7.4, 10 mM MgCl2, 0.01% BSA, 0.0005% Tween 20, 1 mM ATP and 1 &...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 200nMAssay Description:Compounds were added to a 384-well plate. Reaction mixtures contained 10 mM HEPES, pH 7.4, 10 mM MgCl2, 0.01% BSA, 0.0005% Tween 20, 1 mM ATP and 1 &...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 200nMAssay Description:Compounds were added to a 384-well plate. Reaction mixtures contained 10 mM HEPES, pH 7.4, 10 mM MgCl2, 0.01% BSA, 0.0005% Tween 20, 1 mM ATP and 1 &...More data for this Ligand-Target Pair
Ligand Info