BDBM50184872 4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide::4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}-N-(tetrahydro-2H-pyran-4-yl)benzamide::CHEMBL202887::GW-788388
SMILES O=C(NC1CCOCC1)c1ccc(cc1)-c1cc(ccn1)-c1c[nH]nc1-c1ccccn1
InChI Key InChIKey=SAGZIBJAQGBRQA-UHFFFAOYSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50184872
Affinity DataIC50: 446nMAssay Description:Inhibition of TGF-beta1 signaling in human HEK293 cells transfected with luciferase and FAST-2 gene expression vector A3-LUX after 16 hrs by lucifera...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of TbetaR-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Displacement of rhodamine green fluorescently labeled ATP from recombinant GST-ALK5 by FP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.28E+3nMAssay Description:Displacement of rhodamine green fluorescently labeled ATP from recombinant GST-p38alphaMore data for this Ligand-Target Pair