BDBM101649 US9695160, 13::US9796707, Compound 13

SMILES FC(F)(F)c1ccc(N2CCN(Cc3cccnc3)CC2)c(NC(=O)c2ccc(o2)-c2ccncc2)c1

InChI Key InChIKey=UHCHNGAAVWVTIB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 101649   

TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham

US Patent
LigandPNGBDBM101649(US9695160, 13 | US9796707, Compound 13)
Affinity DataIC50:  17.2nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham

US Patent
LigandPNGBDBM101649(US9695160, 13 | US9796707, Compound 13)
Affinity DataIC50:  17nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent