BDBM110163 8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d)
SMILES CCn1c(CCCc2ccccc2)nc2n(CC)c(=O)n(CC)c(=O)c12
InChI Key InChIKey=WAXVCRABQNDHDB-UHFFFAOYSA-N
Data 8 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 110163
Affinity DataKi: 139nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranes in absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 209nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranes in presence of 0.1 mM GTPMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in presence of 0.1 mM GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
North-West University, Private Bag X6001, Potchefstroom 2520, South Africa
North-West University, Private Bag X6001, Potchefstroom 2520, South Africa
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
North-West University, Private Bag X6001, Potchefstroom 2520, South Africa
North-West University, Private Bag X6001, Potchefstroom 2520, South Africa
Affinity DataKi: 2.71E+3nMAssay Description:Displacement of [3H]-NECA from Adenosine A2A receptor in Sprague-Dawley rat striatal membranesMore data for this Ligand-Target Pair