BDBM128117 US8796297, 23
SMILES Nc1nccc(n1)N1CCC2(CNC2)CC1
InChI Key InChIKey=LUKGRPKULAYZKC-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 128117
Affinity DataKi: 12.3nM ΔG°: -10.0kcal/molepH: 7.4 T: 2°CAssay Description:The rat H3 receptor was cloned and expressed in cells, and competition binding assays carried out, according to methods previously described (see Esb...More data for this Ligand-Target Pair
Affinity DataKi: 67.6nM ΔG°: -9.09kcal/molepH: 7.4 T: 2°CAssay Description:The rat H3 receptor was cloned and expressed in cells, and competition binding assays carried out, according to methods previously described (see Esb...More data for this Ligand-Target Pair