BDBM135802 US8853207, Example-82
SMILES COc1ccc(cc1)-c1n[nH]c-2c1Cc1sc(cc-21)-c1ccc(NC(=O)CN2CCCC2)nc1
InChI Key InChIKey=OZSJPXRPIQKJRS-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 135802
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology
US Patent
Development Center For Biotechnology
US Patent
Affinity DataIC50: 12.2nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology
US Patent
Development Center For Biotechnology
US Patent
Affinity DataIC50: 176nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair