BDBM137846 US8871934, 439::US8871934, 474
SMILES Cn1cc(cn1)-c1cc(OCC(=O)N2CC(CO)C2)cc2c1-c1ccccc1C2(O)C(F)(F)F
InChI Key InChIKey=XTCFYLMJVKMCKF-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 137846
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Japan Tobacco
US Patent
Japan Tobacco
US Patent
Affinity DataIC50: 19nMpH: 8.0 T: 2°CAssay Description:The inhibitory action of PDHK activity was indirectly evaluated by performing a kinase reaction in the presence of a test compound and measuring the ...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Japan Tobacco
US Patent
Japan Tobacco
US Patent
Affinity DataIC50: 34nMpH: 8.0 T: 2°CAssay Description:The inhibitory action of PDHK activity was indirectly evaluated by performing a kinase reaction in the presence of a test compound and measuring the ...More data for this Ligand-Target Pair