BDBM148325 US8962637, 137::US8962637, 51

SMILES CN1CCN(Cc2cccc(Nc3ncc4CN(CCc4n3)c3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2)CC1

InChI Key InChIKey=HJRJXYSRPDUZLG-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 148325   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148325(US8962637, 137 | US8962637, 51)
Affinity DataIC50:  7nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148325(US8962637, 137 | US8962637, 51)
Affinity DataIC50:  28nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent