BDBM149696 US8975276, 7

SMILES Cc1ccc(-c2cn3ccc(cc3n2)-c2nc3c(C)ncc(C)n3n2)c(C)c1

InChI Key InChIKey=VVPPGWHZZRJHHT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 149696   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM149696(US8975276, 7)
Affinity DataIC50:  11nMpH: 7.4Assay Description:The PDE10 inhibition assay in 384-well plates was conducted to identify substances for the inhibition of cyclic nucleotide hydrolysis by the PDE10 en...More data for this Ligand-Target Pair
In DepthDetails US Patent