BDBM153271 XZ09
SMILES Cc1ccc(NC(=O)CCC(=O)OCC(=O)c2ccc(cc2)-c2ccccc2)cc1Cl
InChI Key InChIKey=UTUPQHXDVDJNQY-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 153271
Affinity DataIC50: 2.41E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, the compounds in DMSO were added into the LSD1 in the reaction buffer consisting of 50 mM Tris¿HCl, pH 7.5, and 1% DMSO, using Acoustic Tech...More data for this Ligand-Target Pair
Affinity DataIC50: 6.85E+5nMT: 2°CAssay Description:The MAO-A and MAO-B screening biochemical assay was completed by Reaction Biology Corp. with the same assay format with LSD1 assay, and the detailed ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using tyramine as substrate preincubated for 15 mins followed by su...More data for this Ligand-Target Pair
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of human N-terminal KDM1A (151 to 852 residues) using H3 (l to 21 residues)-K4me2 peptide substrate preincubated for 15 mins followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 6.85E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using tyramine as substrate preincubated for 15 mins followed by su...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 2.75E+4nMT: 2°CAssay Description:The MAO-A and MAO-B screening biochemical assay was completed by Reaction Biology Corp. with the same assay format with LSD1 assay, and the detailed ...More data for this Ligand-Target Pair