BDBM154554 (3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)methanone (10)

SMILES CC(C)(C)N1CCN(CC1)C(=O)c1cccc(Br)c1

InChI Key InChIKey=AIAVNBRCOLXLIC-UHFFFAOYSA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 154554   

TargetTP53-binding protein 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPHD finger protein 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMBT domain-containing protein 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPHD finger protein 23(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPHD finger protein 19(Homo sapiens (Human))
University of North Carolina At Chapel Hill

LigandPNGBDBM154554((3-Bromophenyl)(4-(tert-butyl)piperazin-1-yl)metha...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed