BDBM159342 US9034899, 33::US9604960, 33
SMILES Clc1ccc(cc1Cl)C1CNCc2cc(ccc12)-c1cccnn1
InChI Key InChIKey=NRTIHDQHAKWSTG-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 159342
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 6.20nMpH: 7.5 T: 2°CAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 0....More data for this Ligand-Target Pair
Affinity DataIC50: 15.4nMpH: 7.9 T: 2°CAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 0....More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 26nMAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 1....More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 6.20nMAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 0....More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 0....More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 26.4nMpH: 7.5 T: 2°CAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 1....More data for this Ligand-Target Pair